Research Articles

1. Chieh-Hsien Lu, Chung-Wai Shiau, Yung-Chi Chang, Hsiu-Ni Kung, Jui-Ching Wu, Chui-Hian Lim, Hui-Hui Yeo, Han-Chu Chang, Han-Sheng Chien, Sheng-Hsuan Huang, Wei-Kang Hung, Jun-Rong Wei, Hao-Chieh Chiu* (2021 Apr) SC5005 dissipates the membrane potential to kill Staphylococcus aureus persisters without detectable resistance. Journal of Antimicrobial Chemotherapy. DOI: 10.1093/jac/dkab114 (SCI)

2. Tsai-Wen Wan, Yu-Jung Liu, Yu-Ting Wang, Yu-Tzu Lin, Jia-Chuan Hsu, Jui-Chang Tsai, Hao-Chieh Chiu, Po-Ren Hsueh, Wei-Chun Hung, Lee-Jene Teng (2021 Mar) Potentially conjugative plasmids harboring Tn6636, a multidrug-resistant and composite mobile element, in Staphylococcus aureus. Journal of  Microbiology, Immunology and Infection. DOI10.1016/j.jmii.2021.03.003 (SCI)

3. Shiou-Ru Tzeng, Yi-Wei Huang, Yao-Qing Zhang, Ching-Yi Yang, Han-Sheng Chien, Yi-Ru Chen, Sung-Liang Yu, Ching S. Chen, Hao-Chieh Chiu* (2020 Dec) A Celecoxib Derivative Eradicates Antibiotic-Resistant Staphylococcus aureus and Biofilms by Targeting YidC2 Translocase. International Journal of Molecular Sciences. DOI: 10.3390/ijms21239312 (SCI)

4. Ching-Yi Yang, Cheng-Yun Hsu, Chun-Sheng Fang, Chung-Wai Shiau, Ching S. Chen, Hao-Chieh Chiu* (2019 Aug)   Loxapine, an antipsychotic drug, suppresses intracellular multiple-antibiotic-resistant Salmonella enterica serovar Typhimurium in macrophages. Journal of  Microbiology, Immunology and Infection. 52(4):638-647 (SCI)

5. Cheng-Ju Kuo, Sin-Tian Wang, Chia-Mei Lin, Hao-Chieh Chiu, Cheng-Rung Huang, Der-Yen Lee, Geen-Dong Chang, Ting-Chen Chou, Jenn-Wei Chen, Chang-Shi Chen (2018 Mar) A multi-omic analysis reveals the role of fumarate in regulating the virulence of enterohemorrhagic  Escherichia coli. Cell Death and Disease. 7;9(3):381. (SCI)

6. Jung-Chen Su, Yu-Ting Huang, Chang-Shi Chen, Hao-Chieh Chiu*, Chung-Wai Shiau* (2018 Jan) Design and synthesis of malonamide derivatives as antibiotics against methicillin-resistant Staphylococcus aureus. Molecules. 23(1), 27. (SCI)

7. Sung-Pin Tseng, Wei-Chun Hung, Hsiao-Jan Chen, Yu-Tzu Lin, Hung-Sih Jiang, Hao-Chieh Chiu, Po-Ren Hsueh, Lee-Jene Teng, Jui-Chang Tsai (2017 Feb) Effects of toluidine blue O (TBO)-photodynamic inactivation on community-associated methicillin-resistant Staphylococcus aureus isolates. Journal of  Microbiology, Immunology and Infection. 50(1):46-54. (SCI)

8. Kang-Yi Su, Bo-Shiun Yan, Hao-Chieh Chiu, Chong-Jen Yu, So-Yi Chang, Ruwen Jou, Jia-Long Liu, Po-Ren Hsueh, Sung-Liang Yu* (2017 Jan) Rapid Multiplex Detection of M. tuberculosis Complex and Resistant Mutations from Sputum by Mass Spectrometry. Scientific Reports. 7: 41486. (SCI)

9. Cheng-Ju Kuo, Jenn-Wei Chen, Hao-Chieh Chiu, Ching-Hao Teng, Tai-I Hsu, Pei-Jung Lu, Wan-Jr Syu, Sin-Tian Wang, Ting-Chen Chou, Chang-Shi Chen (2016 Aug) Mutation of the enterohemorrhagic Escherichia coli core LPS biosynthesis enzyme RfaD confers hypersusceptibility to host intestinal innate immunity in vivo. Frontiers in Cellular and Infect Microbiology.  6: 82. (SCI)

10. Jung-Chen Su, Ai-Chung Mar, Szu-Hsien Wu, Wei-Tien Tai, Pei-Yi Chu, Chia-Yun Wu, Ling-Ming Tseng, Te-Chang Lee,   Kuen-Feng Chen, Chun-Yu Liu, Hao-Chieh Chiu*, Chung-Wai Shiau* (2016 Jul) Disrupting VEGF-A paracrine and autocrine loops by targeting SHP-1 suppresses triple negative breast cancer metastasis. Scientific Reports. 1;6:28888. (SCI)

11. Han-Chu Chang, Yu-Ting Huang, Chang-Shi Chen, Yi-Wei Chen, Yu-Tsung Huang, Jung-Chen Su, Lee-Jeng Teng, Chung-Wai Shiau, Hao-Chieh Chiu* (2016 Feb.) In Vitro and In Vivo Activity of a Novel Sorafenib Derivative SC5005 against Methicillin-Resistant Staphylococcus aureus. Journal of Antimicrobial Chemotherapy. 71(2):449-59. (SCI)  

12. Hsiao-Jan Chen, Wei-Chun Hung, Yu-Tzu Lin, Jui-Chang Tsai, Hao-Chieh Chiu, Po-Ren Hsueh, Lee-Jene Teng* (2015 Feb) A novel fusidic acid resistance determinant, fusF, in Staphylococcus cohniiJournal of Antimicrobial Chemotherapy. 70(2):416-9 (SCI)

13. Jung-Hsin Lo, Samuel K Kulp, Ching-Shih Chen, Hao-Chieh Chiu* (2014 Dec) Sensitization of Intracellular Salmonella to Aminoglycosides in vitro and in vivo by a Host-Targeted Antimicrobial Agent. Antimicrobial Agents and Chemotherapy. 58(12):7375-82. (SCI)

14. Ya-Luen Yang, Po-Hsien Huang, Hao-Chieh Chiu, Samuel K Kulp, Ching-Shih Chen, Cheng-Ju Kuo, Huan-Da Chen, Chang-Shi Chen* (2013 May) Histone deacetylase inhibitor AR42 regulates telomerase activity in human glioma cells via an Akt-dependent mechanism. Biochemical and Biophysical Research Communications. 24;435(1):107-12. (SCI)

15. Po-Hsien HuangHsiao-Ching Chuang, Chih-Chien ChouHuiling WangSu-Lin LeeHsiao-Ching YangHao-Chieh ChiuNaval KapuriyaDasheng WangSamuel K KulpChing-Shih Chen* (2013 Mar) Vitamin E Facilitates the Inactivation of the Kinase Akt by the Phosphatase PHLPP1. Science Signaling. 6 (267): ra19 (SCI) 

16Ting-Chen Chou#, Hao-Chieh Chiu#, Cheng-Ju Kuo, C.M. Wu, Wan-Jr Syu, Wen-Tai Chiu, Chang-Shi Chen* (2013 Jan) Enterohaemorrhagic Escherichia coli O157:H7 Shiga-like toxin 1 is required for full pathogenicity and activation of the p38 mitogen-activated protein kinase pathway in Caenorhabditis elegans. Cellular Microbiology. 15(1):82-97. (#Equal Contribution) (SCI)

17. Hao-Chieh Chiu, Su-Lin Lee, Naval Kapuriya, Dasheng Wang, Yi-Ru Chen, Sung-Liang Yu, Samuel K. Kulp, Lee-Jene Teng, Ching-Shih Chen* (2012 Aug) Development of novel antibacterial agents against methicillin-resistant Staphylococcus aureusBioorganic & Medicinal Chemistry. 20(15):4653-60. (SCI)

18Hao-Chieh Chiu, Samuel K Kulp, Shilpa Soni, Dasheng Wang, John S Gunn, Larry S Schlesinger, Ching-Shih Chen* (2009 Dec) Eradication of intracellular Salmonella enterica serovar Typhimurium with a small-molecule, host cell-directed agent. Antimicrobial Agents and Chemotherapy. 53:5236-5244. (SCI)

19. Hao-Chieh Chiu, Shilpa Soni, Samuel K Kulp, Heather Curry, Dasheng Wang, John S Gunn, Larry S Schlesinger, Ching-Shih Chen* (2009 Dec) Eradication of intracellular Francisella tularensis in THP-1 human macrophages with a novel autophagy inducing agent. Journal of Biomedical Science. 16:110. (SCI)

20. Hao-Chieh Chiu, Jian Yang, Shilpa Soni, Samuel K Kulp, John S Gunn, Larry S Schlesinger, Ching-Shih Chen* (2009 Jul) Pharmacological exploitation of an off-target antibacterial effect of the cyclooxygenase-2 inhibitor celecoxib against Francisella tularensis. Antimicrobial Agents and Chemotherapy. 53:2998-3002. (SCI)

21. Jui-Wen Huang, Chung-Wai Shiau, Jian Yang, Da-Sheng Wang, Hao-Chieh Chiu, Ching-Yu Chen, Ching-Shih Chen* (2006 Jul) Development of small-molecule cyclin D1-ablative agents. Journal of Medicinal Chemistry. 49:4684-4689. (SCI)

22. Chen-Hua Chuang, Hao-Jie Chiu, Sheng-Chieh Hsu, Jin-Yuan Ho, Wan-Jr Syu* (2006 Jan) Comparison of Tir from enterohemorrahgic and enteropathogenic Escherichia coli strains: two homologues with distinct intracellular properties. Journal of Biomedical Science. 13:73-87. (SCI)

23. Hao-Jie Chiu, Wan-Jr Syu* (2005 Oct) Functional analysis of EspB from enterohaemorrhagic Escherichia coli. Microbiology. 151:3277-3286. (SCI)

24. Hao-Jie Chiu, Wen-Shiun Lin, Wan-Jr Syu* (2003 Sep) Type III secretion of EspB in enterohemorrhagic Escherichia coli O157:H7. Arch Microbiol 180:218-226. (SCI)

Review Articles

1. Hsiao-Jan Chen, Hao-Chieh Chiu, and Lee-Jene Teng* (2012 Mar) Escherichia coli O104:H4. Formosa Journal of Medicine. 16(2): 51-55

2. Hao-Chieh Chiu* and Bo-Shiun Yan (2012 Mar) Tularemia, A Potential Bioterrorism Threat. Formosa Journal of Medicine. 16(2):34-38